Structure-Based Discovery of Negative Allosteric Modulators of the Metabotropic Glutamate Receptor 5

By sjmartinez • November 29, 2022

Kampen S, Rodríguez D, Jørgensen M, Kruszyk-Kujawa M, Huang X, Collins M Jr, Boyle N, Maurel D, Rudling A, Lebon G, Carlsson J. Structure-Based Discovery of Negative Allosteric Modulators of the Metabotropic Glutamate Receptor 5. ACS Chem Biol. 2022 Oct 21;17(10):2744-2752. doi: 10.1021/acschembio.2c00234. Epub 2022 Sep 23. PMID: 36149353; PMCID: PMC9594040.

Tags: Cardiology/Epi, Publications

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